SCHEMBL458979

SCHEMBL458979

O=C=Nc1ccc(C(C2=CCC(N=C=O)(N=C=O)C=C2)c2ccccc2)cc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4647750 0.91
SCHEMBL10436046 0.77
SCHEMBL192102 0.74
SCHEMBL295315 0.73 CYP3A4 (0.47)
SCHEMBL5477781 0.67 ALDH1A1 (0.35)
SCHEMBL93536 0.66 CYP3A4 (0.54)
SCHEMBL11452983 0.66 CYP3A4 (0.39)
SCHEMBL332095 0.65 ALDH1A1 (0.31)
SCHEMBL10539359 0.65 SLC6A2 (0.31)
SCHEMBL10635550 0.65 CYP3A4 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 237 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2009517533-A 2009-04-30 JP claimed
US-20080312403-A1 AROMATIC URETHANE ACRYLATES HAVING A HIGH REFRACTIVE INDEX BAYER MATERIALSCIENCE AG (DE) 2008-12-18 US claimed
EP-1976816-A2 BASE-CATALYZED ALKOXYLATION IN THE PRESENCE OF NON-LINEAR POLYOXYETHYLENE-CONTAINING COMPOUNDS Bayer MaterialScience LLC (US) 2008-10-08 EP claimed
EP-1966275-A1 LONG CHAIN POLYETHER POLYOLS Bayer MaterialScience LLC (US) 2008-09-10 EP claimed
WO-2007117295-A2 BASE-CATALYZED ALKOXYLATION IN THE PRESENCE OF NON-LINEAR POLYOXYETHYLENE-CONTAINING COMPOUNDS BAYER MATERIALSCIENCE LLC (US) 2007-10-18 WO claimed
WO-2007075251-A2 WATER-BLOWN, FLAME RETARDANT RIGID POLYURETHANE FOAM BAYER MATERIALSCIENCE LLC (US) 2007-07-05 WO claimed
WO-2007075482-A1 LONG CHAIN POLYETHER POLYOLS BAYER MATERIALSCIENCE LLC (US) 2007-07-05 WO claimed
EP-1506244-A1 ONE-COMPONENT, WATERBORNE FILM-FORMING COMPOSITION PPG Industries Ohio, Inc. (US) 2005-02-16 EP claimed
US-20040014535-A1 Acid-functional polyurethane and polyurea compositions for golf balls JPMORGAN CHASE BANK, N.A., AS SUCCESSOR ADMINISTRATIVE AGENT 2004-01-22 US claimed
WO-2003099897-A1 ONE-COMPONENT, WATERBORNE FILM-FORMING COMPOSITION PPG INDUSTRIES OHIO, INC. (US) 2003-12-04 WO claimed
US-6610812-B1 Acid functional group based on a carboxylic, sulfonic or phosphonic acid ACUSHNET COMPANY 2003-08-26 US claimed
US-6265468-B1 CROSSLINKED BLEND WITH AROMATIC POLYETHER VIANOVA RESINS, INC. 2001-07-24 US claimed
US-5851667-A Process for production of a composite product CRAY VALLEY S.A. (FR) 1998-12-22 US claimed
EP-0777695-B1 POLYURETHANE COMPOSITIONS HAVING A LOW CONTENT OF MONOMER DIISOCYANATES HENKEL KGAA (DE) 1998-12-02 EP claimed
EP-0172934-A1 Microencapsulated naturally occuring pyrethrins PENNWALT CORPORATION (US) 1986-03-05 EP claimed
US-4497793-A Microencapsulated naturally occuring pyrethrins PENNWALT CORPORATION (US) 1985-02-05 US claimed
US-4110364-A AND BISMALEIIMIDES MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1978-08-29 US claimed
US-20250261306-A1 ADHESIVE-EQUIPPED METAL SUBSTRATE AND LAMINATE ZACROS CORPORATION (JP) 2025-08-14 US disclosed
US-4007239-A CHEMICAL INTERMEDIATE BAYER AKTIENGESELLSCHAFT (DT) 1977-02-08 US disclosed
US-3941849-A CATALYTIC POLYMERIZATION THE GENERAL TIRE & RUBBER COMPANY (US) 1976-03-02 US disclosed