SCHEMBL4590143

SCHEMBL4590143

[CH2]C(CCc1cccc(Cl)c1Cl)SCCCO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.42
PNMT P11086 1/20 0.39
IDO1 P14902 2/20 0.35
ADA P00813 1/20 0.34
TLR8 Q9NR97 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CTSG P08311 1/20 0.32
CMA1 P23946 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
PTPRC P08575 1/20 0.32
PTPRG P23470 1/20 0.32
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C19 P33261 2/20 0.31
CYP2A13 Q16696 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4589469 0.79 TAAR1 (0.41) TAAR1PNMTIDO1ADASLC6A2
SCHEMBL79190 0.76 TAAR1 (0.59) TAAR1PNMTIDO1TLR8CTSG
SCHEMBL29924786 0.72 TAAR1 (0.63) TAAR1PNMTIDO1CTSGCMA1
SCHEMBL2963562 0.72 TAAR1 (0.63) TAAR1PNMTIDO1CTSGCMA1
SCHEMBL4517657 0.70 ADRB2 (0.48) TAAR1PNMTIDO1CTSGCMA1
SCHEMBL4590140 0.70 TAAR1 (0.41) TAAR1PNMTIDO1TLR8KDM4E
SCHEMBL4519480 0.66 PTPRC (0.38) TAAR1PNMTCTSGCMA1PTPRC
SCHEMBL6650913 0.66 TAAR1 (0.59) TAAR1PNMTIDO1KDM4EALDH1A1
SCHEMBL5584502 0.65 TAAR1 (0.63) TAAR1PNMTIDO1KDM4EALDH1A1
SCHEMBL111152 0.64 PNMT (0.62) TAAR1PNMTIDO1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937656-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS BETA 2 ADRENOCEPTOR AGONISTS AstraZeneca AB (SE) 2008-07-02 EP disclosed
WO-2007027134-A1 7-(2-AMINO-1-HYDROXY-ETHYL)-4-HYDROXYBENZOTHIAZOL-2(3H)-ONE-DERIVATIVES AS β2 ADRENOCEPTOR AGONISTS ASTRAZENECA AB (SE) 2007-03-08 WO disclosed