SCHEMBL4590248

SCHEMBL4590248

CC(O)CN1CCC(N2CC(O)CC2=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.36
BLM P54132 1/20 0.36
PARP2 Q9UGN5 1/20 0.35
SLC6A3 Q01959 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HSD11B1 P28845 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573450 0.77 HSD17B10 (0.40) APEX1BLMPARP2POLBGAA
SCHEMBL4573449 0.73 POLB (0.40) APEX1BLMPOLBGAACYP2C19
SCHEMBL4693552 0.72 CHRM2 (0.55) DRD2DRD3
SCHEMBL16311405 0.72 SLC6A3 (0.38) SLC6A3GAADRD2DRD3
SCHEMBL14116233 0.71 SIGMAR1 (0.43) L3MBTL1
SCHEMBL14116439 0.71 SIGMAR1 (0.43) L3MBTL1
SCHEMBL16481901 0.71 POLB (0.61) POLBGAAMEN1KMT2AL3MBTL1
SCHEMBL16481553 0.71 POLB (0.61) POLBGAAMEN1KMT2AL3MBTL1
SCHEMBL18023738 0.70 PARP2 (0.40) PARP2POLBGAAKMT2AL3MBTL1
SCHEMBL31441564 0.68 TP53 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008100621-A2 TETRAHYDRO-PYRAZOLO-PYRIDINE THIOETHER MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. (US) 2008-08-21 WO claimed