SCHEMBL4591082

SCHEMBL4591082

Clc1ccc(-c2cc(Br)cs2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.41
PGR P06401 1/20 0.40
ALAD P13716 1/20 0.39
ALDH1A1 P00352 3/20 0.37
RAB9A P51151 3/20 0.37
MEN1 O00255 2/20 0.37
POLB P06746 2/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
IDO1 P14902 1/20 0.37
PPARG P37231 1/20 0.37
NCOA2 Q15596 1/20 0.37
NCOA1 Q15788 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
AHR P35869 1/20 0.37
NPC1 O15118 2/20 0.37
IKBKB O14920 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598589 0.84 PGR (0.42) PGRALADALDH1A1RAB9AMEN1
SCHEMBL2774954 0.82 CNR1 (0.44) CNR1ALADALDH1A1RAB9AMEN1
SCHEMBL29280044 0.82 BRD4 (0.45) CNR1PGRMAPTIKBKBCYP1A2
SCHEMBL10706711 0.78 HSD17B1 (0.56) MEN1KMT2ACYP3A4CYP2C9HSD17B1
SCHEMBL4590721 0.78 MAPK14 (0.50) PGRALDH1A1RAB9AMEN1MAPT
SCHEMBL3907230 0.77 AR (0.44) CNR1PGRALDH1A1RAB9AMAPT
SCHEMBL28245811 0.77 HSD17B1 (0.46) CNR1ALADALDH1A1MEN1POLB
SCHEMBL27270524 0.77 CNR1 (0.41) CNR1ALADALDH1A1RAB9AMEN1
SCHEMBL10583935 0.77 IKBKB (0.46) CNR1ALADALDH1A1RAB9AMEN1
SCHEMBL4200384 0.77 CNR1 (0.41) CNR1ALADALDH1A1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909775-A2 FORMULATION OF RADIOPROTECTIVE ALPHA, BETA UNSATURATED ARYL SULFONES Onconova Therapeutics, Inc. (US) 2008-04-16 EP disclosed
WO-2007016201-A2 FORMULATION OF RADIOPROTECTIVE α, β UNSATURATED ARYL SULFONES ONCONOVA THERAPEUTICS, INC. (US) 2007-02-08 WO disclosed