SCHEMBL4591121

SCHEMBL4591121

c1ccc(-c2coc(N3CC(c4ncc5cnn(C6CCCCC6)c5n4)C3)n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AURKA O14965 5/20 0.35
CDK1 P06493 5/20 0.35
CCNB1 P14635 4/20 0.35
PDE9A O76083 11/20 0.33
S1PR1 P21453 1/20 0.33
AURKB Q96GD4 1/20 0.33
PDE1C Q14123 2/20 0.33
KCNH2 Q12809 1/20 0.33
PIK3CD O00329 1/20 0.32
RIPK1 Q13546 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4514691 0.81 AURKA (0.41) AURKACDK1CCNB1PDE9AAURKB
SCHEMBL4590637 0.80 SMN1; SMN2 (0.47) KCNH2
SCHEMBL4497277 0.77 PDE9A (0.51) PDE9APDE1C
SCHEMBL4590830 0.72 BCHE (0.45) AURKACDK1CCNB1PDE9APDE1C
SCHEMBL1353660 0.66 CDK4 (0.63) AURKACDK1CCNB1AURKB
SCHEMBL4589851 0.65 LMNA (0.45) AURKACDK1CCNB1PDE9AAURKB
SCHEMBL27156475 0.63 AURKA (0.46) AURKACDK1CCNB1PDE9AAURKB
SCHEMBL8472219 0.62 PDE9A (0.39) AURKACDK1CCNB1PDE9AAURKB
SCHEMBL4497280 0.61 TYK2 (0.50)
SCHEMBL18366799 0.61 AURKA (0.44) AURKACDK1CCNB1PDE9AAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008055959-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-05-15 WO disclosed