SCHEMBL4590830

SCHEMBL4590830

c1ccc2[nH]c(N3CC(c4ncc5cnn(C6CCCCC6)c5n4)C3)nc2c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.45
ACHE P22303 2/20 0.45
PDE10A Q9Y233 1/20 0.45
TRPC3 Q13507 1/20 0.42
HTR3A P46098 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
AURKA O14965 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
PDE9A O76083 3/20 0.38
LMNA P02545 1/20 0.37
KCNH2 Q12809 1/20 0.37
PDE1C Q14123 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4590803 0.80 PDE10A (0.46) BCHEACHEPDE10ATRPC3HTR3A
SCHEMBL4514691 0.80 AURKA (0.41) AURKACDK1CCNB1PDE9AKCNH2
SCHEMBL4510022 0.77 PDE9A (0.53) PDE9APDE1C
SCHEMBL4590637 0.72 SMN1; SMN2 (0.47) TP53MAPTRAB9ALMNAKCNH2
SCHEMBL4591121 0.72 AURKA (0.35) AURKACDK1CCNB1PDE9AKCNH2
SCHEMBL4589851 0.66 LMNA (0.45) MAPTAURKACDK1CCNB1PDE9A
SCHEMBL1353660 0.65 CDK4 (0.63) AURKACDK1CCNB1
SCHEMBL717865 0.65 BCHE (1.00) BCHEACHETRPC3HTR3ATP53
SCHEMBL2241920 0.65 BCHE (1.00) BCHEACHETRPC3HTR3ATP53
SCHEMBL27156475 0.64 AURKA (0.46) AURKACDK1CCNB1PDE9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008055959-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-05-15 WO claimed