SCHEMBL4591568

SCHEMBL4591568

Cc1ccncc1C(=O)ON

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.65
SIRT3 Q9NTG7 1/20 0.65
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
GLA P06280 2/20 0.46
GAA P10253 2/20 0.46
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMYD3 Q9H7B4 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.39
KDM4C Q9H3R0 2/20 0.39
MEN1 O00255 1/20 0.39
KDM6B O15054 1/20 0.39
KDM4A O75164 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4D Q6B0I6 1/20 0.39
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16118580 0.85 ALDH1A1 (0.50) TDP1SIRT3ALDH1A1KDM4EGLA
SCHEMBL1440123 0.83 SIRT3 (0.61) TDP1SIRT3ALDH1A1KDM4EGLA
SCHEMBL30957166 0.83 SIRT3 (0.61) TDP1SIRT3ALDH1A1KDM4EGLA
SCHEMBL5802324 0.81 TDP1 (0.59) TDP1SIRT3ALDH1A1KDM4EGLA
SCHEMBL3964969 0.81 TDP1 (0.65) TDP1SIRT3ALDH1A1KDM4EGLA
SCHEMBL29570949 0.80 SIRT3 (0.58) TDP1SIRT3ALDH1A1NPC1RAB9A
SCHEMBL907851 0.80 SIRT3 (0.58) TDP1SIRT3ALDH1A1NPC1RAB9A
Ethane SCHEMBL28930003 0.79 SIRT3 (0.56) TDP1SIRT3ALDH1A1NPC1RAB9A
SCHEMBL16836475 0.79 ALDH1A1 (0.47) TDP1SIRT3ALDH1A1KDM4EGLA
SCHEMBL28101840 0.79 TDP1 (0.56) TDP1SIRT3ALDH1A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354579-B High-yield synthesis method of methyl 4-aminonicotinate 安徽大学 2024-05-14 CN disclosed
EP-1893603-A1 PIPERIDIN-4-YL-AMIDE DERIVATIVES AND THEIR USE AS SST RECEPTOR SUBTYPE 5 ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2008-03-05 EP disclosed
WO-2006128803-A1 PIPERIDIN-4-YL-AMIDE DERIVATIVES AND THEIR USE AS SST RECEPTOR SUBTYPE 5 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2006-12-07 WO disclosed