SCHEMBL4591683

SCHEMBL4591683

COC(=O)C1CC(=O)c2nc(C)c(C)n2C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.46
KMT2A Q03164 1/20 0.37
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA4 P22748 4/20 0.36
CA6 P23280 4/20 0.36
CA7 P43166 4/20 0.36
CA9 Q16790 4/20 0.36
CA13 Q8N1Q1 4/20 0.36
CA5B Q9Y2D0 3/20 0.35
CA12 O43570 2/20 0.35
CA14 Q9ULX7 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
BUB1 O43683 1/20 0.32
ADORA1 P30542 1/20 0.31
HSP90AA1 P07900 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591532 0.72 BRD4 (0.36) BRD4
SCHEMBL5216737 0.72 LMNA (0.30)
SCHEMBL5217701 0.71 BRD4 (0.42) BRD4
SCHEMBL121399 0.64 BRD4 (1.00) BRD4CA1CA2CA4CA6
SCHEMBL30193882 0.64 BRD4 (1.00) BRD4CA1CA2CA4CA6
SCHEMBL28154981 0.64 BRD4 (0.68) BRD4KMT2ACA1CA2CA4
SCHEMBL16865999 0.63 BRD4 (0.67) BRD4CA1CA2CA4CA6
SCHEMBL18566779 0.62 BRD4 (0.59) BRD4KMT2ACA1CA2CA4
SCHEMBL20875983 0.62 BRD4 (0.64) BRD4KMT2ACA1CA2CA4
SCHEMBL11622652 0.62 MAPT (0.66) BRD4KMT2ACA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899341-A1 SPIRO-IMIDAZNAPHTHYRIDINE DERIVATIVES AS GASTRIC ACID SECRETION INHIBITORS Nycomed GmbH (DE) 2008-03-19 EP disclosed
WO-2006134112-A1 SPIRO-IMIDAZNAPHTHYRIDINE DERIVATIVES AS GASTRIC ACID SECRETION INHIBITORS NYCOMED GMBH (DE) 2006-12-21 WO disclosed