SCHEMBL4592144

SCHEMBL4592144

Cc1cc(C(=O)NC[C@@H]2CCN(C(=O)O)C2)sc1Br

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.40
SMYD3 Q9H7B4 4/20 0.38
KCNH2 Q12809 7/20 0.38
DRD2 P14416 3/20 0.37
DRD4 P21917 3/20 0.37
DRD3 P35462 3/20 0.37
NPC1 O15118 1/20 0.37
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592619 0.88 ACKR3 (0.39) ACKR3SMYD3KCNH2DRD2DRD4
SCHEMBL4592403 0.85 ACKR3 (0.55) ACKR3KDM4EPKM
SCHEMBL3448647 0.85 ACKR3 (0.55) ACKR3KDM4EPKM
SCHEMBL3448652 0.85 ACKR3 (0.55) ACKR3KDM4EPKM
SCHEMBL4592841 0.81 GAA (0.49) ACKR3NPC1KDM4E
SCHEMBL3447821 0.75 ACKR3 (0.56) ACKR3KCNH2KDM4EPKM
SCHEMBL3447823 0.75 ACKR3 (0.56) ACKR3KCNH2KDM4EPKM
SCHEMBL4592664 0.75 ACKR3 (0.56) ACKR3KCNH2KDM4EPKM
SCHEMBL4592552 0.75 F10 (0.52) ACKR3
SCHEMBL8259423 0.75 EP300 (0.47) SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877404-A2 NOVEL CYCLIC AMINES F. Hoffmann-Roche AG (CH) 2008-01-16 EP disclosed
WO-2006114401-A2 NOVEL CYCLIC AMINES F. HOFFMANN-LA ROCHE AG (CH) 2006-11-02 WO disclosed