SCHEMBL4592215

SCHEMBL4592215

NC(=O)OCCc1csc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.53
MTNR1A P48039 1/20 0.47
JUN P05412 1/20 0.46
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
POLB P06746 1/20 0.45
LMNA P02545 1/20 0.44
IDO1 P14902 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.43
TP53 P04637 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
HDAC6 Q9UBN7 2/20 0.42
HDAC1 Q13547 1/20 0.41
MAPT P10636 2/20 0.40
CHRNA7 P36544 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28693243 0.85 CYP2A6 (0.53) CYP2A6MTNR1ACA1CA2POLB
SCHEMBL4592033 0.80 KEAP1 (0.58) CYP2A6MTNR1ACA2SMN1; SMN2MAPT
SCHEMBL8905373 0.80 CYP2A6 (0.58) CYP2A6MTNR1AJUNMAPK8MAPK9
SCHEMBL30138881 0.80 CYP2A6 (0.58) CYP2A6MTNR1AJUNMAPK8MAPK9
SCHEMBL8869956 0.78 CYP2A6 (0.56) CYP2A6MTNR1AJUNMAPK8MAPK9
SCHEMBL27709633 0.78 CYP2A6 (0.45) CYP2A6MTNR1AJUNMAPK8MAPK9
SCHEMBL48674 0.78 POLB (0.64) CYP2A6MTNR1AJUNMAPK8MAPK9
SCHEMBL3070140 0.76 CYP2A6 (0.61) CYP2A6MTNR1AJUNMAPK8MAPK9
SCHEMBL1393298 0.74 CYP2A6 (0.59) CYP2A6MTNR1AJUNMAPK8MAPK9
SCHEMBL8786755 0.74 CYP4F2 (0.60) CYP2A6MTNR1APOLBLMNAIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108264509-B Substituted benzothieno [2,3-c ] tetrahydropyridine derivatives, preparation method and application thereof 复旦大学 2021-05-04 CN disclosed
EP-1904473-A1 BENZOHETEROCYCLYLETHYLCARBOXAMIDE DERIVATIVES Bayer CropScience S.A. (FR) 2008-04-02 EP disclosed
WO-2007006739-A1 BENZOHETEROCYCLYLETHYLCARBOXAMIDE DERIVATIVES BAYER CROPSCIENCE SA (FR) 2007-01-18 WO disclosed