SCHEMBL4592293

SCHEMBL4592293

Nc1c(Br)cc(Cl)cc1CCO

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.34
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 1/20 0.32
ERN1 O75460 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
LMNA P02545 1/20 0.30
GBA1 P04062 1/20 0.30
CYP2D6 P10635 1/20 0.30
CNR1 P21554 1/20 0.30
TBXA2R P21731 1/20 0.30
HRH2 P25021 1/20 0.30
SLC6A4 P31645 1/20 0.30
KCNH2 Q12809 1/20 0.30
HIF1A Q16665 1/20 0.30
TP53 P04637 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19776327 0.84 MCL1 (0.36) MCL1GAAMAPTCYP1A2CYP2C9
SCHEMBL29939894 0.84 MCL1 (0.36) MCL1GAAMAPTCYP1A2CYP2C9
SCHEMBL946031 0.80 HTT (0.38) MCL1GAAMAPTERN1CA1
SCHEMBL27837496 0.80 CYP2D6 (0.45) GAAMAPTCYP1A2CA1CA2
SCHEMBL930175 0.78 ERN1 (0.44) MCL1MAPTCYP1A2CYP2C9ERN1
SCHEMBL28918987 0.78 GAA (0.37) MCL1GAAMAPTERN1CA1
SCHEMBL28060643 0.74 ALDH1A1 (0.39) MAPTCYP1A2LMNAHIF1ACYP3A4
SCHEMBL1639812 0.73 GAA (0.58) MCL1GAAMAPTERN1CA1
SCHEMBL23647915 0.73 ERN1 (0.36) MCL1MAPTCYP1A2CYP2C9ERN1
SCHEMBL3634811 0.72 PYCR1 (0.44) MAPTCYP1A2CYP2C9LMNAHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888538-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-(2-ARYLOXY-ETHYL)-AMINES HAVING AN ACTIVITY ON THE 5-HT RECEPTOR F. Hoffmann-Roche AG (CH) 2008-02-20 EP disclosed
WO-2006117305-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-(2-ARYLOXY-ETHYL)-AMINES HAVING AN ACTIVITY ON THE 5-HT RECEPTOR F. HOFFMANN-LA ROCHE AG (CH) 2006-11-09 WO disclosed