SCHEMBL4593097

SCHEMBL4593097

O=S(=O)(c1ccccc1)C1CNCCN1c1ccc2nc(C(c3ccccc3)C(F)(F)F)[nH]c2c1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.34
SLC6A4 P31645 5/20 0.34
SLC6A3 Q01959 5/20 0.34
CYP2D6 P10635 4/20 0.34
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.33
OPRL1 P41146 1/20 0.32
ACP1 P24666 1/20 0.31
KMT2A Q03164 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
CBFB Q13951 1/20 0.31
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593094 0.77 KMT2A (0.48) LMNASMN1; SMN2ALDH1A1KMT2AKDM4E
SCHEMBL3796418 0.71 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3HTR6
SCHEMBL1887877 0.69 CA12 (0.39) SLC6A2SLC6A4SLC6A3CYP2D6HTR6
SCHEMBL28440794 0.69 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6SMN1; SMN2
SCHEMBL2988535 0.67 S1PR1 (0.42) CYP3A4CYP2C19
SCHEMBL2976716 0.66 BRD4 (0.36) SLC6A2SLC6A4SLC6A3CYP2D6KMT2A
SCHEMBL1890474 0.66 SLC6A4 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6ALDH1A1
SCHEMBL2985975 0.65 ALOX5AP (0.40) SMN1; SMN2MAPT
SCHEMBL1714647 0.64 HTR2C (0.41) ALDH1A1HTR6
SCHEMBL5222798 0.63 KDM4E (0.61) LMNASMN1; SMN2ALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807398-B1 NEW INDOLE OR BENZIMIDAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-06-25 EP disclosed