SCHEMBL1887877

SCHEMBL1887877

O=S(=O)(c1ccccc1)C1CNCCN1c1ccc2occc2c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
SLC6A2 P23975 7/20 0.38
SLC6A4 P31645 7/20 0.38
SLC6A3 Q01959 7/20 0.38
CYP2D6 P10635 3/20 0.38
HTR6 P50406 4/20 0.37
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
KCNH2 Q12809 1/20 0.36
DYRK1A Q13627 1/20 0.36
CHRM5 P08912 2/20 0.35
CTNNB1 P35222 1/20 0.35
WNT3A P56704 1/20 0.35
CHRM1 P11229 1/20 0.35
MMP2 P08253 1/20 0.35
ADAMTS5 Q9UNA0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1890474 0.82 SLC6A4 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL3796418 0.80 SLC6A2 (0.49) SLC6A2SLC6A4SLC6A3HTR6DRD2
SCHEMBL2947702 0.76 SLC6A4 (0.64) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL28440794 0.75 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6HTR6
SCHEMBL2481294 0.71 MAPT (0.64) HTR6
SCHEMBL4593097 0.69 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3CYP2D6HTR6
SCHEMBL30407459 0.69 CHRM2 (0.43) HTR6KCNH2CHRM1
SCHEMBL28061774 0.69 HTR6 (0.42) CA2HTR6KCNH2CHRM1
SCHEMBL1885230 0.68 NR1H4 (0.38) CA2SLC6A4SLC6A3HTR6
SCHEMBL2548093 0.68 DYRK1A (0.58) SLC6A4CYP2D6HTR6DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8575161-B2 Benzofurane, benzothiophene, benzothiazol derivatives as FXR modulators MERCK PATENT GMBH (DE) 2013-11-05 US disclosed
US-20110105475-A1 BENZOFURANE, BENZOTHIOPHENE, BENZOTHIAZOL DERIVATIVES AS FXR MODULATORS MERXCK PATENT GESELLSCHAFT (DE) 2011-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105475-A1 BENZOFURANE, BENZOTHIOPHENE, BENZOTHIAZOL DERIVATIVES AS FXR MODULATORS FXR1, FXR2, NR1H4 CA12 4617/4885CA2 3346/4885SLC6A2 1721/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.