SCHEMBL4595110

SCHEMBL4595110

Fc1cc(C#Cc2ccccc2)cc(Oc2ccccn2)c1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 6/20 0.50
FFAR4 Q5NUL3 1/20 0.46
FFAR1 O14842 1/20 0.38
SCN9A Q15858 1/20 0.38
LTA4H P09960 1/20 0.37
PTGS2 P35354 1/20 0.37
GRM5 P41594 2/20 0.36
NTRK3 Q16288 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30689318 0.83 FFAR4 (0.56) FFAR4SCN9ALTA4HPTGS2GRM5
SCHEMBL4458288 0.76 FFAR4 (0.53) HAO1FFAR4GRM5
SCHEMBL22061563 0.74 KDM4E (0.48) FFAR4LTA4HPTGS2GRM5
SCHEMBL18984715 0.73 MAP4K4 (0.50) FFAR4FFAR1LTA4HPTGS2GRM5
SCHEMBL6369908 0.72 APP (0.60) HAO1FFAR4FFAR1GRM5
SCHEMBL29605037 0.71 SCN9A (0.56) FFAR4SCN9ALTA4HPTGS2
SCHEMBL15954253 0.71 SCN9A (0.56) FFAR4SCN9ALTA4HPTGS2
SCHEMBL22411061 0.71 FFAR4 (0.45) FFAR4SCN9ALTA4HPTGS2
SCHEMBL9368339 0.71 HAO1 (0.45) HAO1FFAR4LTA4HPTGS2GRM5
SCHEMBL13085922 0.70 APP (0.57) HAO1FFAR1LTA4HGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874724-A2 PHENYL ETHYNE COMPOUNDS Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006115895-A2 PHENYL ETHYNE COMPOUNDS MERCK & CO., INC. (US) 2006-11-02 WO disclosed