SCHEMBL4595848

SCHEMBL4595848

CC(C)(C)[C@](CO)(CSCc1ccccc1)NC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.41
LMNA P02545 5/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 3/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
ACE P12821 1/20 0.38
PKM P14618 1/20 0.38
METAP2 P50579 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073210 0.80 CYP3A4 (0.46) CYP2C19LMNAMAPTALDH1A1SMN1; SMN2
SCHEMBL1273081 0.80 CYP3A4 (0.46) CYP2C19LMNAMAPTALDH1A1SMN1; SMN2
SCHEMBL4596217 0.78 NPC1 (0.45) CYP2C19MAPTKDM4EALDH1A1NPC1
SCHEMBL4658500 0.74 KDM4E (0.49) LMNAMAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL9788167 0.73 CYP1A2 (0.41) CYP2C19LMNAALDH1A1HPGDSMN1; SMN2
SCHEMBL8233122 0.73 CYP2C19 (0.45) CYP2C19LMNAMAPTALDH1A1HPGD
SCHEMBL31489064 0.72 CYP1A2 (0.46) CYP2C19LMNAALDH1A1HPGDSMN1; SMN2
SCHEMBL9171687 0.72 CYP2C19 (0.50) CYP2C19LMNAALDH1A1HPGDSMN1; SMN2
SCHEMBL13696274 0.71 CYP2C19 (0.46) CYP2C19LMNAALDH1A1HPGDSMN1; SMN2
SCHEMBL8233124 0.71 PPARG (0.45) CYP2C19LMNAMAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874768-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113837-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed