SCHEMBL4595950

SCHEMBL4595950

NC(=O)C(Sc1ccccc1)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.43
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
POLB P06746 2/20 0.37
MAPK1 P28482 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
CPA1 P15085 1/20 0.37
CES1 P23141 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
PKM P14618 1/20 0.35
MAPT P10636 2/20 0.35
PARP1 P09874 1/20 0.34
TSHR P16473 1/20 0.34
RECQL P46063 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686346 0.74 EPHX1 (0.45) EPHX1LMNASMN1; SMN2L3MBTL1POLB
SCHEMBL820641 0.74 CYP2C19 (0.45) EPHX1LMNASMN1; SMN2L3MBTL1POLB
SCHEMBL5902536 0.71 EPHX1 (0.42) EPHX1LMNASMN1; SMN2L3MBTL1POLB
SCHEMBL2311192 0.71 EPHX1 (0.66) EPHX1LMNASMN1; SMN2L3MBTL1PKM
SCHEMBL27618189 0.70 MEN1 (0.43) LMNASMN1; SMN2CES1CYP2C19CYP1A2
SCHEMBL11371564 0.70 FFAR1 (0.39) LMNASMN1; SMN2L3MBTL1POLBMAPK1
SCHEMBL6796251 0.69 EPHX1 (0.71) EPHX1LMNASMN1; SMN2L3MBTL1POLB
SCHEMBL8659778 0.69 POLB (0.46) LMNASMN1; SMN2L3MBTL1POLBMAPK1
SCHEMBL585643 0.69 SMN1; SMN2 (0.39) LMNASMN1; SMN2L3MBTL1POLBMAPK1
SCHEMBL1483540 0.68 EPHX1 (0.46) EPHX1LMNASMN1; SMN2L3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008100621-A2 TETRAHYDRO-PYRAZOLO-PYRIDINE THIOETHER MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. (US) 2008-08-21 WO disclosed