SCHEMBL4596446

SCHEMBL4596446

O=C1CCOc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=C1CCSc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=C1CN=Cc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 8/20 0.43
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
AKT1 P31749 3/20 0.32
CA9 Q16790 1/20 0.32
TDP2 O95551 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
CDK2 P24941 2/20 0.31
CDK1 P06493 1/20 0.31
KIT P10721 1/20 0.31
KDR P35968 1/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
PDE3B Q13370 2/20 0.31
PDE3A Q14432 2/20 0.31
MMP8 P22894 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4897633 0.80 KIF11 (0.57) KIF11AKT1CA9TDP2CDK2
SCHEMBL4595242 0.80 KIF11 (0.64) KIF11CYP11B1CYP11B2CA9TDP2
SCHEMBL4596143 0.79 KIF11 (0.66) KIF11CYP11B1CYP11B2AKT1TDP2
SCHEMBL4596854 0.72 KIF11 (0.47) KIF11AKT1TDP2CDK2CDK1
SCHEMBL4596430 0.71 KIF11 (0.59) KIF11CYP11B1CYP11B2TDP2TRPV1
SCHEMBL4596362 0.68 KIF11 (0.61) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL4596493 0.66 NOTUM (0.47) KIF11CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL4595131 0.64 KIF11 (0.50) KIF11CYP11B1CYP11B2AKT1TDP2
SCHEMBL15964654 0.64 KIF11 (0.48) KIF11TRPV1
SCHEMBL2632666 0.64 HDAC1 (0.53) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP claimed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO claimed
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed