SCHEMBL4595131

SCHEMBL4595131

O=C1CCCc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=C1CCc2cc(-c3ccc(C(F)(F)F)cc3)cc(F)c2N1.O=C1CCc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=C1COc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=C1CSc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 15/20 0.50
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
AKT1 P31749 1/20 0.34
TDP2 O95551 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4888035 0.74 KIF11 (0.86) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4893178 0.74 KIF11 (0.63) KIF11CYP11B1CYP11B2TDP2
SCHEMBL4596430 0.74 KIF11 (0.59) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4596362 0.73 KIF11 (0.61) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4888861 0.72 KIF11 (0.86) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4596393 0.71 KIF11 (0.39) KIF11CYP11B1CYP11B2
SCHEMBL1396616 0.71 KIF11 (1.00) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4596868 0.70 KIF11 (0.65) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4596019 0.69 KIF11 (0.44) KIF11PDE3BPDE3AAKT1
SCHEMBL4595242 0.68 KIF11 (0.64) KIF11PDE3BPDE3ACYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP claimed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO claimed