SCHEMBL4597033

SCHEMBL4597033

O=c1c(NCc2cccc(O)c2)c(Nc2ccc3ncsc3c2)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.52
PLK1 P53350 1/20 0.44
ROCK1 Q13464 5/20 0.43
ROCK2 O75116 4/20 0.43
CHEK2 O96017 4/20 0.43
PRKACA P17612 4/20 0.43
RPS6KB1 P23443 4/20 0.43
AKT1 P31749 4/20 0.43
GSK3B P49841 4/20 0.43
RPS6KA3 P51812 4/20 0.43
PRKG1 Q13976 4/20 0.43
PKN2 Q16513 4/20 0.43
CDC42BPA Q5VT25 4/20 0.43
HIPK4 Q8NE63 4/20 0.43
AURKB Q96GD4 4/20 0.43
CHEK1 O14757 3/20 0.43
AKT2 P31751 3/20 0.43
CLK2 P49760 3/20 0.43
PRKAA1 Q13131 3/20 0.43
PRKG2 Q13237 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4598968 0.91 RPS6KB1 (0.43) KDRROCK1ROCK2CHEK2PRKACA
SCHEMBL4597939 0.85 KDR (0.48) KDRPLK1ROCK1ROCK2CHEK2
SCHEMBL30513613 0.79 SYK (0.48) KDRPLK1GSK3BCLK2CLK4
SCHEMBL28639993 0.79 SYK (0.48) KDRPLK1GSK3BCLK2CLK4
SCHEMBL4905846 0.79 MAPKAPK2 (0.61) PLK1ROCK1ROCK2CHEK2GSK3B
SCHEMBL4897789 0.79 MAPKAPK2 (0.61) PLK1ROCK1ROCK2CHEK2GSK3B
SCHEMBL4906887 0.78 MAPKAPK2 (0.54) KDRROCK1ROCK2CHEK2PRKACA
SCHEMBL4596911 0.78 NAMPT (0.47) KDRROCK1ROCK2CHEK2PRKACA
SCHEMBL4597203 0.77 KMT2A (0.46) KDRROCK1ROCK2CHEK2PRKACA
SCHEMBL4902096 0.77 NOTUM (0.43) KDRROCK1ROCK2CHEK2PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed