SCHEMBL30513613

SCHEMBL30513613

O=c1c(NCc2ccccn2)c(Nc2ccc3ncsc3c2)c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.48
KDR P35968 4/20 0.48
PLK1 P53350 1/20 0.47
PTPN11 Q06124 1/20 0.46
DYRK3 O43781 2/20 0.42
CLK1 P49759 2/20 0.42
CLK2 P49760 2/20 0.42
CLK3 P49761 2/20 0.42
GSK3B P49841 2/20 0.42
DYRK1A Q13627 2/20 0.42
DYRK2 Q92630 2/20 0.42
CLK4 Q9HAZ1 2/20 0.42
DYRK4 Q9NR20 2/20 0.42
DYRK1B Q9Y463 2/20 0.42
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
MAP3K8 P41279 1/20 0.41
INSR P06213 3/20 0.41
TEK Q02763 3/20 0.41
PDGFRB P09619 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28639993 1.00 SYK (0.48) SYKKDRPLK1PTPN11DYRK3
SCHEMBL30513611 0.91 PTPN11 (0.46) SYKKDRPLK1PTPN11MAOA
SCHEMBL28632683 0.91 PTPN11 (0.46) SYKKDRPLK1PTPN11MAOA
SCHEMBL28651320 0.80 PTPN11 (0.41) PTPN11GSK3BMAOAMAOBABCB1
SCHEMBL30513609 0.80 PTPN11 (0.41) PTPN11GSK3BMAOAMAOBABCB1
SCHEMBL28644056 0.80 PTPN11 (0.48) PTPN11GSK3BMAOAMAOBMAP3K8
SCHEMBL4597033 0.79 KDR (0.52) SYKKDRPLK1DYRK3CLK2
SCHEMBL28637102 0.78 MAOA (0.63) GSK3BCLK4MAOAMAOBABCB1
SCHEMBL30513601 0.78 MAPT (0.56) PTPN11CLK2GSK3BDYRK1ACLK4
SCHEMBL28641831 0.78 MAPT (0.56) PTPN11CLK2GSK3BDYRK1ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759549-B 3-substituted amino-4- ((substituted pyridinyl) amino) cyclobut-3-ene-1, 2-dione compounds 中国医学科学院药物研究所 2023-07-28 CN disclosed