SCHEMBL4597774

SCHEMBL4597774

Cc1cccc([C@@H]2CN(C3CCNCC3)C(=O)N2)c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.54
HTR2A P28223 2/20 0.41
HTR2B P41595 2/20 0.41
ADRB1 P08588 1/20 0.40
TP53 P04637 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PBRM1 Q86U86 3/20 0.36
NSD3 Q9BZ95 1/20 0.36
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36
PARP1 P09874 1/20 0.36
HTR6 P50406 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608509 1.00 HTR2C (0.54) HTR2CHTR2AHTR2BADRB1TP53
SCHEMBL4598053 0.84 SLC18A3 (0.44) HTR2CHTR2AHTR2BTP53KMT2A
SCHEMBL2604304 0.84 SLC18A3 (0.44) HTR2CHTR2AHTR2BTP53KMT2A
SCHEMBL4596627 0.81 HTR2C (0.41) HTR2CHTR2AHTR2BADRB1MEN1
SCHEMBL3248250 0.76 CALCRL (0.38) HTR2CHTR2AHTR2BTP53MEN1
SCHEMBL3247820 0.76 MEN1 (0.37) HTR2CHTR2AHTR2BTP53MEN1
Trifluoroacetic Acid SCHEMBL3253412 0.75 CALCRL (0.43) HTR2CHTR2AHTR2BNSD3PARP1
SCHEMBL5573761 0.73 CCR5 (0.51) HTR2C
SCHEMBL5573756 0.73 CCR5 (0.51) HTR2C
SCHEMBL4597778 0.72 HTR2C (0.52) HTR2CHTR2AHTR2BADRB1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed