SCHEMBL4597833

SCHEMBL4597833

O=Cc1ccc(Oc2ccc(C(=O)O)cc2)nc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.66
L3MBTL1 Q9Y468 3/20 0.66
KDM4E B2RXH2 2/20 0.66
OPRM1 P35372 7/20 0.49
OPRD1 P41143 7/20 0.49
OPRK1 P41145 6/20 0.49
POLB P06746 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.48
PARP10 Q53GL7 2/20 0.47
PARP3 Q9Y6F1 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MAPT P10636 1/20 0.46
SRD5A2 P31213 1/20 0.46
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
GRIN1 Q05586 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3698466 0.91 ALDH1A1 (0.57) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL3696133 0.87 PARP10 (0.67) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL31621360 0.85 ALDH1A1 (0.81) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL4596521 0.84 KDM4E (0.65) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL31556429 0.82 ALDH1A1 (0.71) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL510519 0.82 ALDH1A1 (0.71) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL8016831 0.82 KDM4E (0.66) ALDH1A1L3MBTL1KDM4EPOLBNPC1
SCHEMBL4597726 0.81 KDM4E (0.60) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL3692143 0.81 PARP10 (0.67) ALDH1A1L3MBTL1KDM4EOPRM1OPRD1
SCHEMBL1448984 0.80 ALDH1A1 (0.76) ALDH1A1KDM4EPARP10PARP3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed