SCHEMBL4598116

SCHEMBL4598116

COC(=O)C1=C(c2ccc(COCC3CC3)cc2)CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.42
CHRM5 P08912 4/20 0.41
CHRM1 P11229 4/20 0.41
CHRM2 P08172 3/20 0.41
CHRM4 P08173 3/20 0.41
CHRM3 P20309 3/20 0.41
ESR2 Q92731 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN6 P29350 1/20 0.39
SLC6A2 P23975 1/20 0.38
GPR119 Q8TDV5 3/20 0.38
HDAC1 Q13547 2/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
YAP1 P46937 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597030 0.90 ESR2 (0.40) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL9350724 0.84 GPR119 (0.47) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL1750511 0.83 ESR2 (0.53) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL9350854 0.82 DDB1 (0.39) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL5274358 0.81 NR1H2 (0.45) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL1750649 0.80 CHRM5 (0.48) CHRM5CHRM1CHRM2CHRM4CHRM3
SCHEMBL951478 0.80 NR1H2 (0.47) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL3197517 0.80 SLC6A3 (0.54) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL6418231 0.79 CHRM5 (0.59) NR1H2CHRM5CHRM1CHRM2CHRM4
SCHEMBL5941814 0.77 CHRM5 (0.45) NR1H2CHRM5CHRM1CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1908471-A1 Tetrahydropyridines as renin inhibitors Speedel Experimenta AG (CH) 2008-04-09 EP disclosed