SCHEMBL4598309

SCHEMBL4598309

CN(C)CCNC(=O)CC(Nc1c(Nc2ccc3nc[nH]c3c2)c(=O)c1=O)c1cccc(O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.40
POLB P06746 1/20 0.40
MAPKAPK2 P49137 2/20 0.38
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
QPCT Q16769 4/20 0.37
NAMPT P43490 2/20 0.36
EPHX1 P07099 1/20 0.36
CYP2C9 P11712 1/20 0.36
PDGFRA P16234 1/20 0.36
PRKCA P17252 1/20 0.36
ROCK1 Q13464 1/20 0.36
RPS6KA1 Q15418 1/20 0.36
AURKB Q96GD4 1/20 0.36
CSNK1G1 Q9HCP0 1/20 0.36
MELK Q14680 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
SYK P43405 1/20 0.35
P2RY14 Q15391 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14066740 0.94 MAPKAPK2 (0.38) MAPK1POLBMAPKAPK2AURKARPS6KB1
SCHEMBL14066741 0.82 HPGD (0.38) MAPK1POLBMAPKAPK2CYP2C9PDGFRA
SCHEMBL4908818 0.78 MAPKAPK2 (0.42) MAPK1POLBMAPKAPK2QPCTNAMPT
SCHEMBL4910847 0.77 MAPKAPK2 (0.42) MAPK1POLBMAPKAPK2QPCTCYP2C9
SCHEMBL4599129 0.76 MAPKAPK2 (0.45) MAPK1MAPKAPK2QPCTCYP2C9PDGFRA
SCHEMBL4906181 0.76 MAPKAPK2 (0.40) MAPK1POLBMAPKAPK2QPCTCYP2C9
SCHEMBL4598396 0.73 QPCT (0.49) POLBMAPKAPK2QPCT
SCHEMBL4898077 0.72 MAPKAPK2 (0.37) MAPK1MAPKAPK2CYP2C9PDGFRAPRKCA
SCHEMBL4598398 0.71 CXCR2 (0.41) MAPK1MAPKAPK2CYP2C9PDGFRAPRKCA
SCHEMBL4596962 0.71 MAPKAPK2 (0.61) MAPK1MAPKAPK2CYP2C9PDGFRAPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed