SCHEMBL4598401

SCHEMBL4598401

O=c1c(NCc2cccc(O)c2)c(NCc2ccc3nc[nH]c3c2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.47
ABL1 P00519 1/20 0.44
NAMPT P43490 1/20 0.44
QPCT Q16769 5/20 0.42
F2 P00734 1/20 0.42
PRSS1 P07477 1/20 0.42
POLB P06746 1/20 0.42
IP6K1 Q92551 1/20 0.42
AURKA O14965 2/20 0.42
AURKB Q96GD4 2/20 0.42
NLRP3 Q96P20 1/20 0.41
PDGFRB P09619 1/20 0.41
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
ATM Q13315 1/20 0.40
RPS6KB1 P23443 1/20 0.40
P2RY14 Q15391 1/20 0.40
ALPL P05186 1/20 0.40
ALPI P09923 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4898767 0.90 RPS6KB1 (0.40) KDRABL1NAMPTIP6K1AURKA
SCHEMBL4596911 0.90 NAMPT (0.47) KDRABL1NAMPTQPCTIP6K1
SCHEMBL4905587 0.83 ROCK1 (0.48) KDRABL1NAMPTQPCTIP6K1
SCHEMBL4905562 0.82 KDR (0.44) KDRABL1QPCTF2PRSS1
SCHEMBL4905113 0.82 AURKB (0.39) KDRABL1NAMPTQPCTPOLB
SCHEMBL4907244 0.81 GSK3B (0.41) KDRABL1IP6K1AURKAAURKB
SCHEMBL4598825 0.79 QPCT (0.47) KDRNAMPTQPCTF2PRSS1
SCHEMBL4900151 0.79 MAPKAPK2 (0.47) KDRAURKBRPS6KB1
SCHEMBL4907742 0.79 MAPKAPK2 (0.47) KDRAURKBRPS6KB1
SCHEMBL14066719 0.77 IP6K1 (0.55) KDRNAMPTQPCTIP6K1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910312-A1 QUADRATIC ACID II DERIVATIVES Merck Patent GmbH (DE) 2008-04-16 EP claimed
WO-2007014608-A1 QUADRATIC ACID II DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-08 WO claimed