SCHEMBL4598586

SCHEMBL4598586

Brc1ccc(-c2[c]scc2Br)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 1/20 0.36
CYP2A6 P11509 1/20 0.35
MAPT P10636 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
IDO1 P14902 1/20 0.33
CA12 O43570 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
NPC1 O15118 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ALAD P13716 1/20 0.32
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
LTA4H P09960 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7253183 0.78
SCHEMBL4591911 0.64 ALDH1A1 (0.39) ALDH1A1MAPK1CYP2A6MAPTRAB9A
SCHEMBL68094 0.63 ALDH1A1 (0.73) ALDH1A1MAPK1CYP2A6MAPTRAB9A
SCHEMBL12302096 0.63 ALDH1A1 (0.73) ALDH1A1MAPK1CYP2A6MAPTRAB9A
SCHEMBL1673427 0.63 ALDH1A1 (0.73) ALDH1A1MAPK1CYP2A6MAPTRAB9A
Water SCHEMBL3824552 0.60 ALDH1A1 (0.69) ALDH1A1MAPK1CYP2A6MAPTRAB9A
SCHEMBL1255210 0.60 ALDH1A1 (0.69) ALDH1A1MAPK1CYP2A6MAPTRAB9A
SCHEMBL21518323 0.60 ALDH1A1 (0.69) ALDH1A1MAPK1CYP2A6MAPTRAB9A
Bromide SCHEMBL29066324 0.60 ALDH1A1 (0.69) ALDH1A1MAPK1CYP2A6MAPTRAB9A
Hydrogen Sulfide SCHEMBL4123828 0.60 ALDH1A1 (0.69) ALDH1A1MAPK1CYP2A6MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909775-A2 FORMULATION OF RADIOPROTECTIVE ALPHA, BETA UNSATURATED ARYL SULFONES Onconova Therapeutics, Inc. (US) 2008-04-16 EP disclosed
WO-2007016201-A2 FORMULATION OF RADIOPROTECTIVE α, β UNSATURATED ARYL SULFONES ONCONOVA THERAPEUTICS, INC. (US) 2007-02-08 WO disclosed