SCHEMBL4598855

SCHEMBL4598855

COc1cccc2c1C1Nc3cc(C#N)ccc3C(C)(C)C1CS2

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.33
AR P10275 3/20 0.33
NR3C2 P08235 2/20 0.33
NR3C1 P04150 1/20 0.33
PGR P06401 1/20 0.33
ESRRA P11474 7/20 0.32
ACHE P22303 2/20 0.31
GSK3B P49841 2/20 0.31
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
ESRRB O95718 1/20 0.30
ESR1 P03372 1/20 0.30
ESRRG P62508 1/20 0.30
ESR2 Q92731 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4555983 1.00 SNCA (0.33) SNCAARNR3C2NR3C1PGR
SCHEMBL4815232 0.83 CREBBP (0.37)
SCHEMBL4629098 0.80 AR (0.34) ARNR3C2NR3C1PGRACHE
SCHEMBL4570013 0.80 AR (0.34) ARNR3C2NR3C1PGRACHE
SCHEMBL4813632 0.80 CREBBP (0.35) PGR
SCHEMBL4565983 0.78
SCHEMBL4814159 0.77 HDAC4 (0.33)
SCHEMBL4445324 0.77 HDAC4 (0.33)
SCHEMBL4866034 0.77 NR3C1 (0.35) ARNR3C2NR3C1PGRESRRA
SCHEMBL4816048 0.77 KMT2A (0.34) SNCAARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907395-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-04-09 EP disclosed
WO-2007002867-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2007-01-04 WO disclosed