SCHEMBL4599794

SCHEMBL4599794

O=CC(F)c1ccc(Br)s1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
DAO P14920 2/20 0.33
WRN Q14191 1/20 0.33
HSD17B2 P37059 1/20 0.32
TOP2A P11388 1/20 0.31
TOP2B Q02880 1/20 0.31
GSK3B P49841 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
PKM P14618 1/20 0.30
HPGD P15428 1/20 0.30
MAPK1 P28482 1/20 0.30
NTSR1 P30989 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21495021 0.77 CES2 (0.35) CES2CES1DAOWRNHSD17B2
SCHEMBL193502 0.77 CES2 (0.35) CES2CES1DAOWRNHSD17B2
SCHEMBL7069962 0.75 CES2 (0.34) CES2CES1DAOWRNHSD17B2
SCHEMBL4173122 0.69
SCHEMBL5147505 0.67 CES2 (0.36) CES2CES1DAOWRNHSD17B2
SCHEMBL1066616 0.67
SCHEMBL2505676 0.66 WRN (0.38) CES2CES1DAOWRNHSD17B2
SCHEMBL680628 0.66
SCHEMBL7449320 0.64 GSK3B (0.33) WRNGSK3B
SCHEMBL16799715 0.64 DAO (0.39) CES2CES1DAOWRNKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910307-A1 PYRAZOLE BASED LXR MODULATORS Exelixis, Inc. (US) 2008-04-16 EP disclosed
WO-2007002559-A1 PYRAZOLE BASED LXR MODULATORS EXELIXIS, INC. (US) 2007-01-04 WO disclosed