SCHEMBL7069962

SCHEMBL7069962

O=CC(Cl)c1ccc(Br)s1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
GSK3B P49841 2/20 0.33
DAO P14920 1/20 0.33
WRN Q14191 1/20 0.33
HSD17B2 P37059 1/20 0.32
TOP2A P11388 1/20 0.31
TOP2B Q02880 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
PKM P14618 1/20 0.30
HPGD P15428 1/20 0.30
MAPK1 P28482 1/20 0.30
NTSR1 P30989 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL193502 0.77 CES2 (0.35) CES2CES1GSK3BDAOWRN
SCHEMBL7067216 0.77 GABBR2 (0.40) GSK3BDAOWRNTOP2ATOP2B
SCHEMBL21495021 0.77 CES2 (0.35) CES2CES1GSK3BDAOWRN
SCHEMBL4599794 0.75 CES2 (0.34) CES2CES1GSK3BDAOWRN
SCHEMBL7449320 0.72 GSK3B (0.33) GSK3BWRN
SCHEMBL7068733 0.69 GSK3B (0.44) GSK3BDAOKDM4EALDH1A1LMNA
SCHEMBL28723184 0.69 GSK3B (0.35) GSK3B
SCHEMBL371534 0.69 GSK3B (0.35) GSK3B
SCHEMBL4173122 0.69
SCHEMBL1163934 0.68 CES2 (0.41) CES2CES1GSK3BDAOWRN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055479-A1 COMPOUNDS AND THEIR THERAPEUTIC USE RELATED TO THE PHOSPHORYLATING ACTIVITY OF THE ENZYME GSK-3 CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS (ES) 2003-07-10 WO disclosed