SCHEMBL4600240

SCHEMBL4600240

[AsH2]c1ccccc1-c1nc2ncccc2o1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.68
ALDH1A1 P00352 4/20 0.66
GAA P10253 3/20 0.66
MAPT P10636 3/20 0.66
HPGD P15428 3/20 0.66
HSD17B10 Q99714 2/20 0.66
NPC1 O15118 8/20 0.54
RAB9A P51151 7/20 0.54
SMN1; SMN2 Q16637 5/20 0.52
TP53 P04637 1/20 0.46
ALOX12 P18054 1/20 0.46
HAVCR2 Q8TDQ0 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SIRT1 Q96EB6 2/20 0.44
F2 P00734 1/20 0.43
F10 P00742 1/20 0.43
F7 P08709 1/20 0.43
F3 P13726 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13522986 0.81 NPC1 (0.69) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL9646773 0.81 KDM4E (1.00) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL220575 0.81 KDM4E (0.68) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL9867464 0.81 KDM4E (0.68) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL11645613 0.81 KDM4E (0.68) KDM4EALDH1A1GAAMAPTHPGD
Iodide SCHEMBL11648822 0.79 KDM4E (0.97) KDM4EALDH1A1GAAMAPTHPGD
Iodide SCHEMBL11648817 0.79 KDM4E (0.97) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL26833315 0.79 ALDH1A1 (1.00) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL11640732 0.77 KDM4E (0.62) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL9868647 0.77 KDM4E (0.62) KDM4EALDH1A1GAAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910384-A1 IMIDAZO [2,1-B]THIAYOLE DERIVATIVES AS SIRTUIN MODULATING COMPOUNDS Sirtris Pharmaceuticals, Inc. (US) 2008-04-16 EP disclosed
WO-2007019344-A1 IMIDAZO [2,1-B] THIAYOLE DERIVATIVES AS SIRTUIN MODULATING COMPOUNDS SIRTRIS PHARMACEUTICALS, INC. (US) 2007-02-15 WO disclosed