SCHEMBL4600592

SCHEMBL4600592

O=C(O)[C@H]1CN(C(=O)O)C[C@@H]1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GABRR1 P24046 3/20 0.39
GRM4 Q14833 4/20 0.33
CYP2C19 P33261 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
GRM8 O00222 1/20 0.33
GRM6 O15303 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
GRM2 Q14416 1/20 0.33
GABRR2 P28476 1/20 0.33
PEPD P12955 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17747644 0.88 GABRR1 (0.37) GABRR1GRM4CYP2C19MEN1ALDH1A1
SCHEMBL3183946 0.85 GABRR1 (0.33) GABRR1
SCHEMBL15194169 0.85 GABRR1 (0.33) GABRR1
SCHEMBL15193898 0.85 GABRR1 (0.33) GABRR1
SCHEMBL3197102 0.85 GABRR1 (0.33) GABRR1
SCHEMBL17632223 0.83 CHRNB2 (0.35)
SCHEMBL26615125 0.83 GABRR1 (0.48) GABRR1GRM4CYP2C19MEN1ALDH1A1
SCHEMBL6791728 0.83 GABRR1 (0.48) GABRR1GRM4CYP2C19MEN1ALDH1A1
SCHEMBL21682481 0.83 GABRR1 (0.48) GABRR1GRM4CYP2C19MEN1ALDH1A1
SCHEMBL28866517 0.83 CHRNB2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240118281-A1 ANTICANCER COMPOUNDS AND USES THEREOF UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-04-11 US disclosed
US-20160137639-A1 TRIAZOLE-ISOXAZOLE COMPOUND AND MEDICAL USE THEREOF JAPAN TOBACCO INC. (JP) 2016-05-19 US disclosed
EP-1877404-A2 NOVEL CYCLIC AMINES F. Hoffmann-Roche AG (CH) 2008-01-16 EP disclosed
WO-2006114401-A2 NOVEL CYCLIC AMINES F. HOFFMANN-LA ROCHE AG (CH) 2006-11-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240118281-A1 ANTICANCER COMPOUNDS AND USES THEREOF MKI67, TP53, PCNA GABRR1 4380/4885GRM4 4695/4885CYP2C19 4312/4885
US-20160137639-A1 TRIAZOLE-ISOXAZOLE COMPOUND AND MEDICAL USE THEREOF CYP3A7, CYP2C19, CYP3A5 GABRR1 435/4885GRM4 2373/4885CYP2C19 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.