SCHEMBL4601158

SCHEMBL4601158

CC(C)(C)OC(=O)Nc1cc(Cl)c(F)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 5/20 0.44
CYP17A1 P05093 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
RXFP1 Q9HBX9 1/20 0.37
HTT P42858 2/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
KCNQ4 P56696 1/20 0.36
KCNQ5 Q9NR82 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ATR Q13535 1/20 0.36
EGFR P00533 1/20 0.35
AURKB Q96GD4 1/20 0.35
RORC P51449 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29697261 0.87 CYP17A1 (0.44) CYP17A1CA12CA1CA2CA9
SCHEMBL22990771 0.87 CYP17A1 (0.44) CYP17A1CA12CA1CA2CA9
SCHEMBL29840249 0.83 AAK1 (0.46) AAK1CYP17A1CA12CA1CA2
SCHEMBL3568182 0.83 AAK1 (0.40) AAK1CYP17A1CA12CA1CA2
SCHEMBL29236468 0.83 CYP17A1 (0.42) AAK1CYP17A1CA12CA1CA2
SCHEMBL30947444 0.83 CYP17A1 (0.42) AAK1CYP17A1CA12CA1CA2
SCHEMBL27214502 0.82 CA12 (0.42) AAK1CA12CA1CA2CA9
SCHEMBL2294920 0.82 ATR (0.40) CYP17A1CA12CA1CA2CA9
SCHEMBL15834220 0.82 ALDH1A1 (0.45) AAK1MEN1KMT2A
SCHEMBL31736070 0.81 AAK1 (0.52) AAK1CYP17A1RXFP1HTTKCNQ4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896396-A1 ANTHRANILIC ACID DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-03-12 EP disclosed
WO-2006134040-A1 ANTHRANILIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-12-21 WO disclosed