SCHEMBL4602736

SCHEMBL4602736

CC1(NC(=O)c2ccc(NC(=O)Cc3ccc(Br)c(Oc4cc(Cl)cc(C#N)c4)c3F)c(Cl)c2)C(=O)C[SH4]C1=O

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.35
KCNH2 Q12809 2/20 0.32
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2950902 0.85 CYP3A4 (0.37) CYP3A4KCNH2CYP2C9CYP2C19
SCHEMBL3913666 0.84 KCNH2 (0.35) CYP3A4KCNH2CYP2C9CYP2C19
SCHEMBL2945296 0.84 CYP3A4 (0.37) CYP3A4KCNH2
SCHEMBL2942807 0.84 KCNH2 (0.35) CYP3A4KCNH2
SCHEMBL2950737 0.84 DGAT2 (0.41)
SCHEMBL4605798 0.83 CYP3A4 (0.36) CYP3A4KCNH2CYP2C9CYP2C19
SCHEMBL2949608 0.82 CYP3A4 (0.36) CYP3A4KCNH2CYP2C9CYP2C19
SCHEMBL2950724 0.81 CYP3A4 (0.38) CYP3A4KCNH2CYP2C9CYP2C19
SCHEMBL2944695 0.81 CYP3A4 (0.38) CYP3A4KCNH2CYP2C9CYP2C19
SCHEMBL2951433 0.81 CYP3A4 (0.36) CYP3A4KCNH2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940782-A1 N-PHENYL PHENYLACETAMIDE NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INIHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2008-07-09 EP claimed
WO-2007045572-A1 N-PHENYL PHENYLACETAMIDE NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INIHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2007-04-26 WO claimed