SCHEMBL4603071

SCHEMBL4603071

CCOC(=O)c1nc(-c2ccccc2Cl)n(-c2ccc(OCc3ccccc3)cc2)c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.57
CACNA2D1 P54289 1/20 0.47
L3MBTL1 Q9Y468 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
PKM P14618 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 1/20 0.45
HSP90AA1 P07900 1/20 0.45
KMT2A Q03164 1/20 0.45
CNR2 P34972 3/20 0.44
LMNA P02545 1/20 0.43
PPARG P37231 1/20 0.43
CHRNA7 P36544 1/20 0.43
TP53 P04637 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAOB P27338 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4902164 0.91 CNR1 (0.54) CNR1CACNA2D1L3MBTL1NPC1RAB9A
SCHEMBL3093294 0.91 CNR1 (0.70) CNR1CNR2
SCHEMBL4905590 0.90 CNR1 (0.60) CNR1CACNA2D1L3MBTL1NPC1RAB9A
4-Imidazolecarboxylic Acid SCHEMBL4617313 0.82 CNR1 (0.48) CNR1CACNA2D1L3MBTL1NPC1RAB9A
SCHEMBL4904252 0.82 CNR1 (0.66) CNR1CNR2
SCHEMBL4617309 0.80 CNR1 (0.47) CNR1CACNA2D1L3MBTL1NPC1RAB9A
SCHEMBL3080647 0.80 CNR1 (0.74) CNR1L3MBTL1NPC1RAB9ACNR2
SCHEMBL6332827 0.77 CNR1 (0.53) CNR1NPC1RAB9AKMT2ACNR2
SCHEMBL4616359 0.77 CNR1 (0.48) CNR1CNR2CHRNA7
SCHEMBL739526 0.75 CNR1 (0.64) CNR1NPC1RAB9ACNR2GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080306115-A1 Midazole-4-Carboxamide Derivatives For Use As Cb1 Modulators ASTRAZENECA AB (SE) 2008-12-11 US disclosed
EP-1940820-A1 MIDAZOLE-4-CARBOXAMIDE DERIVATIVES FOR USE AS CB MODULATORS AstraZeneca AB (SE) 2008-07-09 EP disclosed
WO-2007031721-A1 MIDAZOLE-4-CARBOXAMIDE DERIVATIVES FOR USE AS CB MODULATORS ASTRAZENECA AB (SE) 2007-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306115-A1 Midazole-4-Carboxamide Derivatives For Use As Cb1 Modulators CNR2, CNR1, FAAH CNR1 2/4885CACNA2D1 1007/4885L3MBTL1 4710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.