SCHEMBL4604450

SCHEMBL4604450

CCOC(=O)Oc1ccc2[nH]cnc2c1Cl

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
MEN1 O00255 1/20 0.40
CASP1 P29466 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TSHR P16473 1/20 0.39
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
KDM5B Q9UGL1 1/20 0.35
CUL4A Q13619 1/20 0.35
TYMS P04818 1/20 0.35
PARP1 P09874 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4603481 0.99 KDM4E (0.39) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL4604974 0.81 PARP1 (0.46) KDM4EHPGDHSD17B10MEN1KMT2A
SCHEMBL4907498 0.78 KDM4E (0.44) KDM4EALDH1A1HPGDHSD17B10MEN1
Hydrochloric Acid SCHEMBL4914353 0.77 KDM4E (0.43) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL20472000 0.74 BRD4 (0.47) ALDH1A1MEN1KMT2APKM
SCHEMBL4777812 0.73 TP53 (0.39) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL4604722 0.70 CA2 (0.44) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL9542969 0.70 KDM4E (0.40) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL4607622 0.68 LMNA (0.40) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL4089116 0.68 SMN1; SMN2 (0.52) KDM4EALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed