SCHEMBL4605047

SCHEMBL4605047

COc1ccc(CNC(Oc2cccc3[nH]c4ccccc4c23)C(C)O)c(OC)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.45
DNM1 Q05193 2/20 0.45
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
MAPT P10636 3/20 0.43
DRD2 P14416 3/20 0.43
TLR4 O00206 2/20 0.43
ADRB1 P08588 2/20 0.43
ADRB3 P13945 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SLC22A2 O15244 1/20 0.43
SLC22A1 O15245 1/20 0.43
MLNR O43193 1/20 0.43
NR1I2 O75469 1/20 0.43
KCNK2 O95069 1/20 0.43
ABCB11 O95342 1/20 0.43
APP P05067 1/20 0.43
ABCB1 P08183 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4457452 0.80 ADRB2 (0.53) ADRB2DNM1BCHEACHEMAPT
SCHEMBL2995900 0.78 ADRB3 (0.66) ADRB2DNM1MAPTDRD2TLR4
SCHEMBL2995641 0.78 ADRB3 (0.66) ADRB2DNM1MAPTDRD2TLR4
SCHEMBL2993362 0.78 ADRB3 (0.66) ADRB2DNM1MAPTDRD2TLR4
SCHEMBL789339 0.78 ADRB2 (0.63) ADRB2DNM1BCHEACHEMAPT
SCHEMBL6507182 0.77 ADRB2 (0.54) ADRB2DNM1BCHEACHEMAPT
SCHEMBL4608341 0.75 ADRB2 (0.53) ADRB2DNM1BCHEACHEMAPT
SCHEMBL9621537 0.74 ADRB2 (0.55) ADRB2DNM1BCHEACHEMAPT
Hydrochloric Acid SCHEMBL6553108 0.74 ADRB3 (0.45) ADRB2DNM1TLR4ADRB1ADRB3
SCHEMBL4727264 0.72 ADRB2 (0.50) ADRB2DNM1BCHEACHEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP disclosed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO disclosed