SCHEMBL6507182

SCHEMBL6507182

CCCNC(Oc1cccc2[nH]c3ccccc3c12)C(C)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.54
DNM1 Q05193 2/20 0.54
ADRB3 P13945 5/20 0.45
TLR4 O00206 4/20 0.45
DRD2 P14416 3/20 0.45
MAPT P10636 2/20 0.45
KCNH2 Q12809 2/20 0.45
KDM4E B2RXH2 1/20 0.45
SLC22A2 O15244 1/20 0.45
SLC22A1 O15245 1/20 0.45
MLNR O43193 1/20 0.45
NR1I2 O75469 1/20 0.45
KCNK2 O95069 1/20 0.45
ABCB11 O95342 1/20 0.45
APP P05067 1/20 0.45
ABCB1 P08183 1/20 0.45
ADRB1 P08588 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
ADORA3 P0DMS8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4457452 0.85 ADRB2 (0.53) ADRB2DNM1ADRB3TLR4DRD2
SCHEMBL789339 0.85 ADRB2 (0.63) ADRB2DNM1ADRB3TLR4DRD2
SCHEMBL4608341 0.84 ADRB2 (0.53) ADRB2DNM1ADRB3TLR4DRD2
SCHEMBL9621537 0.83 ADRB2 (0.55) ADRB2DNM1ADRB3TLR4DRD2
SCHEMBL4727264 0.81 ADRB2 (0.50) ADRB2DNM1ADRB3TLR4DRD2
SCHEMBL5320295 0.80 HTR1B (0.49) ADRB2ADRB3KCNH2KDM4ESLC22A1
SCHEMBL7702692 0.79 ADRB3 (0.67) ADRB2DNM1ADRB3ADRB1
SCHEMBL4607220 0.79 ADRB3 (0.48) ADRB2DNM1ADRB3TLR4DRD2
SCHEMBL7701306 0.78 ADRB3 (0.68) ADRB2DNM1ADRB3ADRB1UTS2R
SCHEMBL7438512 0.77 ADRB2 (0.61) ADRB2DNM1ADRB3TLR4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005099699-A1 COMBINATION OF (S)-AMLODIPINE AND A BETA-BLOCKER, AND METHODS FOR REDUCING HYPERTENSION SEPRACOR INC. (US) 2005-10-27 WO disclosed