SCHEMBL4606730

SCHEMBL4606730

CC(C)(CNC(=O)c1ccccc1O)Cc1cnccc1C=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 3/20 0.40
HPGD P15428 2/20 0.40
ESRRG P62508 1/20 0.39
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NAAA Q02083 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NLRP1 Q9C000 1/20 0.35
CA1 P00915 2/20 0.35
CA9 Q16790 2/20 0.35
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4606675 0.91 KDM4E (0.40) KMT2AALDH1A1KDM4EMEN1HPGD
SCHEMBL4607563 0.79 KDM4E (0.41) KMT2AALDH1A1KDM4EMEN1HPGD
SCHEMBL4607163 0.79 MAPK1 (0.49) KMT2AALDH1A1KDM4EMEN1HPGD
SCHEMBL9676593 0.75 HPGD (0.51) KMT2AALDH1A1KDM4EMEN1HPGD
SCHEMBL4608634 0.73 HPGD (0.47) KMT2AALDH1A1KDM4EMEN1HPGD
SCHEMBL4610234 0.73 ESRRG (0.47) KMT2AALDH1A1HPGDESRRGRAB9A
SCHEMBL17205426 0.72 CHRNB2 (0.44) KMT2AALDH1A1KDM4EMEN1HPGD
SCHEMBL4606799 0.72 ACHE (0.52) KMT2AMEN1POLB
SCHEMBL4607660 0.72 ACHE (0.52) KMT2AMEN1POLB
SCHEMBL4072495 0.69 CYP2C9 (0.35) ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440976-B1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production BOEHRINGER INGELHEIM PHARMA (DE) 2008-07-23 EP disclosed
EP-1440976-A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production Boehringer Ingelheim Pharma GmbH & Co.KG (DE) 2004-07-28 EP disclosed
EP-0927192-B1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION BOEHRINGER INGELHEIM PHARMA (DE) 2004-05-12 EP disclosed
EP-0927192-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1999-07-07 EP disclosed
WO-1998011128-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1998-03-19 WO disclosed