SCHEMBL4606783

SCHEMBL4606783

CCN(CC)CCOc1c(C)[nH]c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
KDM4E B2RXH2 2/20 0.48
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTT P42858 2/20 0.44
HTR6 P50406 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
CYP1A2 P05177 1/20 0.42
LTA4H P09960 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTR1A P08908 1/20 0.42
AHR P35869 1/20 0.42
MPO P05164 1/20 0.42
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
ALK Q9UM73 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3556246 0.85 HTR6 (0.56) TSHRHTR2AHTR2CHTTHTR6
SCHEMBL13496586 0.81 KDM4E (0.41) TSHRKDM4EHTR2CALDH1A1MAPT
SCHEMBL1827429 0.81 SMN1; SMN2 (0.46) TSHRKDM4EALDH1A1MAPTCYP1A2
SCHEMBL3462132 0.80 HTR2A (0.44) TSHRKDM4EHTR2AHTR2CHTT
SCHEMBL5746662 0.74 HTR1B (0.51) KDM4EHTR2AHTR2CHTTHTR6
SCHEMBL20970934 0.74 HTR6 (0.71) TSHRKDM4EHTR2AHTR2CHTT
SCHEMBL29536604 0.74 HTR6 (0.71) TSHRKDM4EHTR2AHTR2CHTT
SCHEMBL14141474 0.73 HTR6 (0.65) TSHRKDM4EHTR2AHTR2CHTT
SCHEMBL853973 0.71 HTR2A (0.47) KDM4EHTR2AHTR2CHTTALDH1A1
SCHEMBL5749322 0.70 ABCG2 (0.59) TSHRKDM4EHTR2AHTR2CHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1947085-A1 Substituted indole sulfonamide compounds, their preparation and use as medicaments Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed
EP-1947085-A1 Substituted indole sulfonamide compounds, their preparation and use as medicaments Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed