SCHEMBL4606846

SCHEMBL4606846

CC(C)S(=O)(=O)NC1CCCC1c1ccc(NC(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 13/20 0.74
GRIA2 P42262 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4606850 1.00 GRIA4 (0.74) GRIA4GRIA2
SCHEMBL4607083 0.90 GRIA4 (0.60) GRIA4GRIA2
SCHEMBL4606949 0.90 GRIA4 (0.60) GRIA4GRIA2
SCHEMBL4606558 0.90 GRIA4 (0.60) GRIA4GRIA2
SCHEMBL4606652 0.90 GRIA4 (0.60) GRIA4GRIA2
SCHEMBL4607162 0.89 GRIA4 (0.59) GRIA4GRIA2
SCHEMBL4605406 0.89 GRIA4 (0.59) GRIA4GRIA2
SCHEMBL4607600 0.89 GRIA4 (0.70) GRIA4GRIA2
SCHEMBL4607075 0.89 GRIA4 (0.70) GRIA4GRIA2
SCHEMBL4605760 0.88 GRIA4 (0.58) GRIA4GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP claimed
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP disclosed
US-6639107-B1 Potentiating glutamate receptor function ELI LILLY AND COMPANY 2003-10-28 US disclosed
EP-1246797-A1 CYCLOPENTYL SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2002-10-09 EP disclosed
WO-2001042203-A1 CYCLOPENTYL SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-06-14 WO disclosed