SCHEMBL4607016

SCHEMBL4607016

Cc1cc(O)c(C)c(S)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.65
SELL P14151 1/20 0.50
SELP P16109 1/20 0.50
SELE P16581 1/20 0.50
TRPA1 O75762 2/20 0.40
ALDH1A1 P00352 6/20 0.39
CYP3A4 P08684 2/20 0.37
MAPT P10636 4/20 0.37
POLB P06746 3/20 0.37
KMT2A Q03164 3/20 0.37
GAA P10253 3/20 0.37
APEX1 P27695 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MPI P34949 1/20 0.37
RECQL P46063 1/20 0.37
PIM1 P11309 3/20 0.34
LMNA P02545 4/20 0.33
TP53 P04637 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
DAO P14920 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11600377 0.93 ACHE (0.56) ACHESELLSELPSELETRPA1
SCHEMBL20788821 0.80 ACHE (0.40) ACHESELLSELPSELEALDH1A1
SCHEMBL69718 0.80 ACHE (1.00) ACHESELLSELPSELETRPA1
SCHEMBL63242 0.79 ACHE (0.43) ACHESELLSELPSELECYP3A4
SCHEMBL11330631 0.76 ACHE (0.46) ACHESELLSELPSELETRPA1
SCHEMBL11027321 0.75 SELL (0.50) ACHESELLSELPSELETRPA1
SCHEMBL1402361 0.72 RAPGEF4 (0.39) ACHEALDH1A1MAPTGAAKDM4E
SCHEMBL16528140 0.72 ACHE (0.72) ACHESELLSELPSELETRPA1
SCHEMBL205747 0.72 ACHE (0.72) ACHESELLSELPSELETRPA1
Formaldehyde SCHEMBL10878707 0.72 ACHE (0.82) ACHESELLSELPSELETRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2838891-B1 AROMATIC RING COMPOUND AS GHRELIN O-ACYLTRANSFERASE INHIBITOR TAKEDA PHARMACEUTICALS CO (JP) 2017-08-02 EP disclosed
CN-104254525-B aromatic ring compound TAKEDA PHARMACEUTICAL CO.,LTD. (JP) 2016-05-25 CN disclosed
US-9238639-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-01-19 US disclosed
CN-104254525-A Aromatic ring compound TAKEDA PHARMACEUTICAL 2014-12-31 CN disclosed
EP-1945620-A2 COMPOUNDS AND COMPOSITIONS AS PPAR MODULATORS IRM LLC (BM) 2008-07-23 EP disclosed
WO-2007056366-A2 COMPOUNDS AND COMPOSITIONS AS PPAR MODULATORS IRM LLC (BM) 2007-05-18 WO disclosed