SCHEMBL4607295

SCHEMBL4607295

CC(C)S(=O)(=O)N[C@@H]1CCC[C@H]1c1ccc(-c2cccc(NS(C)(=O)=O)c2)cc1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 7/20 0.73
KCNH2 Q12809 5/20 0.73
GRIA4 P48058 11/20 0.60
KDM1A O60341 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14141327 1.00 GRIA2 (0.73) GRIA2KCNH2GRIA4KDM1A
SCHEMBL4605918 1.00 GRIA2 (0.73) GRIA2KCNH2GRIA4KDM1A
SCHEMBL7250833 0.85 GRIA2 (0.74) GRIA2KCNH2GRIA4KDM1A
SCHEMBL4607084 0.85 GRIA2 (0.74) GRIA2KCNH2GRIA4KDM1A
SCHEMBL7250835 0.85 GRIA2 (0.74) GRIA2KCNH2GRIA4KDM1A
SCHEMBL4606632 0.85 GRIA4 (0.71) GRIA2KCNH2GRIA4
SCHEMBL4604598 0.85 KDM1A (0.58) GRIA2KCNH2GRIA4KDM1A
SCHEMBL4604595 0.85 KDM1A (0.58) GRIA2KCNH2GRIA4KDM1A
SCHEMBL4956505 0.84 GRIA2 (1.00) GRIA2KCNH2KDM1A
SCHEMBL5185917 0.84 GRIA2 (0.71) GRIA2KCNH2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP claimed
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP disclosed