SCHEMBL4607462

SCHEMBL4607462

CN(CC(=O)O)c1ccccc1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
ALOX15 P16050 1/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TSHR P16473 2/20 0.46
TP53 P04637 1/20 0.46
PTPN1 P18031 5/20 0.43
KDM4E B2RXH2 4/20 0.41
TDP1 Q9NUW8 3/20 0.41
HPGD P15428 2/20 0.41
POLB P06746 2/20 0.41
LMNA P02545 1/20 0.41
GLA P06280 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
HMGB1 P09429 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14399058 0.87 PTPN1 (0.46) ALDH1A1ALOX15GAAMAPTSMN1; SMN2
SCHEMBL31084573 0.85 ALDH1A1 (0.50) ALDH1A1ALOX15GAAMAPTSMN1; SMN2
SCHEMBL26423787 0.83 ALDH1A1 (0.48) ALDH1A1ALOX15GAAMAPTSMN1; SMN2
SCHEMBL20274405 0.82 EGFR (0.41) ALDH1A1GAAMAPTSMN1; SMN2TSHR
SCHEMBL3948272 0.81 NOTUM (0.50) ALDH1A1TP53KDM4ETDP1LMNA
SCHEMBL30580347 0.81 TDP1 (0.56) ALDH1A1ALOX15GAAMAPTSMN1; SMN2
SCHEMBL129880 0.81 TDP1 (0.56) ALDH1A1ALOX15GAAMAPTSMN1; SMN2
SCHEMBL31357954 0.80 ALDH1A1 (0.45) ALDH1A1ALOX15GAAMAPTSMN1; SMN2
SCHEMBL3276453 0.80 ABCC1 (0.53) ALDH1A1ALOX15TSHRPTPN1HPGD
SCHEMBL1051805 0.80 PTPN1 (0.46) ALDH1A1ALOX15GAAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5942372-A COMPRISED A SPECTRAL SENSITIZER THAT SENSITIZES IN THE ULTRAVIOLET OR VISIBLE REGIONS OF THE SPECTRUM AND AN N-ARYL POLYCARBOXYLIC ACID CO-INITIATOR; VERY HIGH PHOTOSPEED AND VERY GOOD SHELF-LIFE IN COMPUTER-TO-PLATE SYSTEMS KODAK POLYCHROME GRAPHICS, LLC (US) 1999-08-24 US claimed
US-5914215-A ELEMENT COMPRISING SUPPORT HAVING PHOTOIMAGEABLE, RADIATION SENSITIVE LAYER COMPRISING UNSATURATED COMPOUND, PHOTOINITIATOR SYSTEM COMPRISING SENSITIZER SENSITIZING IN ULTRAVIOLET OR VISIBLE REGION OF SPECTRUM, CO-INITIATOR KODAK POLYCHROME GRAPHIC, LLC (US) 1999-06-22 US claimed
EP-0783577-B1 CHIMERIC RECEPTORS AND METHODS FOR IDENTIFYING COMPOUNDS ACTIVE AT METABOTROPIC GLUTAMATE RECEPTORS AND THE USE OF SUCH COMPOUNDS IN THE TREATMENT OF NEUROLOGICAL DISORDERS AND DISEASES ASTRAZENECA AB (SE) 2008-07-09 EP disclosed
EP-0882065-B1 NOVEL HUMAN METABOTROPIC GLUTAMATE RECEPTOR NPS PHARMA INC (US) 2007-08-08 EP disclosed
EP-1687402-A4 CHIMERIC METABOTROPIC GLUTAMATE RECEPTORS AND USES THEREOF NPS PHARMA INC (US) 2007-08-01 EP disclosed
US-7241863-B2 Human metabotropic glutamate receptor NPS PHARMACEUTICALS, INC. (US) 2007-07-10 US disclosed
US-7232467-B2 Dyeing hair with capped diazonium compound; intense, striking coloration; light, shampoo and rub fastness; storage stability; nondamaging, nonstaining CIBA SPECIALTY CHEMICALS CORPORATION (US) 2007-06-19 US disclosed
US-7232467-B2 Dyeing hair with capped diazonium compound; intense, striking coloration; light, shampoo and rub fastness; storage stability; nondamaging, nonstaining CIBA SPECIALTY CHEMICALS CORPORATION (US) 2007-06-19 US disclosed
US-7229479-B2 Method of coloring porous material CIBA SPECIALTY CHEMICALS CORPORATION (US) 2007-06-12 US disclosed
US-7229479-B2 Method of coloring porous material CIBA SPECIALTY CHEMICALS CORPORATION (US) 2007-06-12 US disclosed
US-7223295-B2 Dyeing hair with capped diazonium compound; intense, striking coloration; light, shampoo and rub fastness; storage stability; nondamaging, nonstaining CIBA SPECIALTY CHEMICALS CORPORATION (US) 2007-05-29 US disclosed
US-5821030-A DIRECT DIGITAL EXPOSURE; HIGH WRITING SPEED; ADHESION; ANTIFOGGING AGENTS; SHELF LIFE; USING A POLYCARBOXYLIC ACID IN THE PHOTOPOLYMERIZATION INITIATOR SYSTEM AND A BASIC COMPOUND IN THE OXYGEN BARRIER LAYER KODAK POLYCHROME GRAPHICS (US) 1998-10-13 US disclosed
US-5776655-A CONTAINING PHOTOPOLYMER EASTMAN KODAK COMPANY (US) 1998-07-07 US disclosed
WO-1997048724-A2 HUMAN METABOTROPIC GLUTAMATE RECEPTOR NPS PHARMACEUTICALS, INC. (US) 1997-12-24 WO disclosed
EP-0795790-A2 Peel-developable lithographic printing plate EASTMAN KODAK COMPANY (US) 1997-09-17 EP disclosed
EP-0783577-A1 CHIMERIC RECEPTORS AND METHODS FOR IDENTIFYING COMPOUNDS ACTIVE AT METABOTROPIC GLUTAMATE RECEPTORS AND THE USE OF SUCH COMPOUNDS IN THE TREATMENT OF NEUROLOGICAL DISORDERS AND DISEASES NPS PHARMACEUTICALS, INC. (US) 1997-07-16 EP disclosed
US-5629354-A Photopolymerization initiator system comprising a spectral sensitizer and a polycarboxylic acid co-initiator EASTMAN KODAK COMPANY (US) 1997-05-13 US disclosed
WO-1997005252-A2 CHIMERIC RECEPTORS AND METHODS FOR IDENTIFYING COMPOUNDS ACTIVE AT METABOTROPIC GLUTAMATE RECEPTORS AND THE USE OF SUCH COMPOUNDS IN THE TREATMENT OF NEUROLOGICAL DISORDERS AND DISEASES NPS PHARMACEUTICALS, INC. (US) 1997-02-13 WO disclosed
EP-0730201-A1 Sensitized photopolymerizable compositions and use thereof in lithographic printing plates EASTMAN KODAK COMPANY (US) 1996-09-04 EP disclosed
WO-1996005818-A1 METHODS AND COMPOUNDS ACTIVE AT METABOTROPIC GLUTAMATE RECEPTORS USEFUL FOR TREATMENT OF NEUROLOGICAL DISORDERS AND DISEASES NPS PHARMACEUTICALS, INC. (US) 1996-02-29 WO disclosed