SCHEMBL4607944

SCHEMBL4607944

CC(O)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)C(F)(F)F

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 20/20 0.74
PDK2 Q15119 20/20 0.74
PDK3 Q15120 20/20 0.74
PDK4 Q16654 20/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6568377 0.91 PDK1 (0.74) PDK1PDK2PDK3PDK4
SCHEMBL4608424 0.86 PDK1 (0.63) PDK1PDK2PDK3PDK4
SCHEMBL25026296 0.85 ALDH1A1 (0.55) PDK1PDK2PDK3PDK4
SCHEMBL6348275 0.85 PDK1 (1.00) PDK1PDK2PDK3PDK4
SCHEMBL31053831 0.85 ALDH1A1 (0.55) PDK1PDK2PDK3PDK4
SCHEMBL4610340 0.85 PDK1 (0.73) PDK1PDK2PDK3PDK4
SCHEMBL6348342 0.84 PDK1 (0.76) PDK1PDK2PDK3PDK4
SCHEMBL6348339 0.84 PDK1 (0.76) PDK1PDK2PDK3PDK4
SCHEMBL4608920 0.83 PDK1 (0.59) PDK1PDK2PDK3PDK4
SCHEMBL4608925 0.83 PDK1 (0.59) PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1059927-B1 CHEMICAL COMPOUNDS AND THEIR USE TO ELEVATE PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 2008-07-30 EP disclosed