SCHEMBL4609399

SCHEMBL4609399

FC(F)(F)c1ccccc1-c1cccc2c1C[C]O2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.36
HSD11B1 P28845 2/20 0.35
AR P10275 1/20 0.35
SCN9A Q15858 2/20 0.35
PSMB8 P28062 1/20 0.34
EPHX2 P34913 1/20 0.33
CNR2 P34972 1/20 0.33
SLC9A1 P19634 1/20 0.33
GALR1 P47211 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDK2 Q15119 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
TRPA1 O75762 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596282 0.75 AR (0.37) NOTUMHSD11B1ARSCN9APSMB8
SCHEMBL4609397 0.73 NOTUM (0.37) NOTUMHSD11B1ARSCN9APSMB8
SCHEMBL197671 0.71 HSD11B1 (0.56) NOTUMHSD11B1ARPSMB8ALDH1A1
SCHEMBL8022901 0.69 HSD11B1 (0.54) NOTUMHSD11B1ARPSMB8ALDH1A1
Hydrochloric Acid SCHEMBL29010139 0.69 HSD11B1 (0.54) NOTUMHSD11B1ARPSMB8ALDH1A1
SCHEMBL4595505 0.68 AR (0.34) NOTUMHSD11B1ARSCN9APSMB8
SCHEMBL4223592 0.67 HTR2C (0.40) NOTUMHSD11B1ARSCN9AALDH1A1
SCHEMBL16193459 0.66 CES1 (0.40) NOTUMHSD11B1ARSCN9APSMB8
SCHEMBL18646126 0.66 GALR1 (0.41) NOTUMHSD11B1ARSCN9APSMB8
SCHEMBL15540806 0.66 HSD11B1 (0.47) NOTUMHSD11B1ARPSMB8GALR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed