SCHEMBL4609561

SCHEMBL4609561

[CH2]Oc1cnc(F)c(-c2ccc(Cl)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA7 P36544 1/20 0.39
MAP4K4 O95819 4/20 0.36
CYP1A2 P05177 1/20 0.36
KCNH2 Q12809 1/20 0.36
MINK1 Q8N4C8 1/20 0.36
TNIK Q9UKE5 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MEN1 O00255 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KMT2A Q03164 2/20 0.34
PTGS2 P35354 1/20 0.34
LTA4H P09960 1/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4609563 0.84 NPSR1 (0.46) CHRNB4CHRNA3CHRNA7MAP4K4CYP1A2
SCHEMBL411023 0.79 BACE1 (0.44) MAP4K4CYP1A2KCNH2MINK1TNIK
SCHEMBL3143008 0.76 CHRNB4 (0.39) CHRNB4CHRNA3CHRNA7MAP4K4KCNH2
Hydrochloric Acid SCHEMBL3773488 0.75 CHRNB4 (0.39) CHRNB4CHRNA3CHRNA7MAP4K4KCNH2
Hydrochloric Acid SCHEMBL3773493 0.74 CHRNB4 (0.40) CHRNB4CHRNA3CHRNA7KCNH2FFAR4
SCHEMBL3137211 0.70 FFAR4 (0.38) CHRNB4CHRNA3CHRNA7MAP4K4FFAR4
SCHEMBL3137206 0.70 FFAR4 (0.38) CHRNB4CHRNA3CHRNA7MAP4K4FFAR4
SCHEMBL16879689 0.65 GSTP1 (0.55) CYP1A2NPSR1MEN1NPC1RAB9A
SCHEMBL3875252 0.65 CYP11B2 (0.55) CYP1A2PTGS2
SCHEMBL3550859 0.63 AHR (0.42) MAP4K4CYP1A2KCNH2MINK1TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-A1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Les Laboratoires Servier (FR) 2008-10-15 EP disclosed
WO-2007085750-A1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2007-08-02 WO disclosed