SCHEMBL4609747

SCHEMBL4609747

O=C(O)N1CCC(S(=O)(=O)NCc2ccccc2)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
CA2 P00918 3/20 0.45
CA1 P00915 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
TACR3 P29371 1/20 0.43
CA12 O43570 2/20 0.42
CA7 P43166 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL56220 0.83 STS (0.56) MEN1KMT2ACA1CA12CA7
SCHEMBL11953320 0.80 SMN1; SMN2 (0.61) MEN1KMT2ACA2CA1NPSR1
SCHEMBL55795 0.78 STS (0.61) MEN1KMT2ACA1CA12CA7
SCHEMBL3811125 0.77 CA12 (0.59) KMT2ACA2CA1CA12CA7
SCHEMBL11946070 0.77 NSD2 (0.51) CA2CA1CA12CA7CA14
SCHEMBL65669 0.77 NPY5R (0.39) MEN1KMT2ANPSR1
SCHEMBL14721003 0.76 CXCR4 (0.58) MEN1KMT2ANPSR1HDAC3HDAC4
SCHEMBL27890613 0.75 NSD2 (0.53) CA2CA1CA12CA7CA14
SCHEMBL1189971 0.74 ACHE (0.60) MEN1KMT2ANPSR1
SCHEMBL16269315 0.74 ACHE (0.60) MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948597-A1 DERIVATIVES FOR MODULATION OF ION CHANNELS Vertex Pharmaceuticals Incorporated (US) 2008-07-30 EP disclosed
WO-2007050522-A1 DERIVATIVES FOR MODULATION OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-03 WO disclosed