SCHEMBL4611181

SCHEMBL4611181

CN(C)C(=O)C1(N2CCCC2)CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CA2 P00918 1/20 0.33
CHKA P35790 1/20 0.33
KDM4E B2RXH2 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3898636 0.98 CA2 (0.36) CYP1A2CA2CHKAKDM4EKMT2A
Hydrochloric Acid SCHEMBL4609226 0.97 CA2 (0.35) CYP1A2CA2CHKA
SCHEMBL14434750 0.84 CA2 (0.36) CYP1A2CA2CHKAKMT2A
SCHEMBL6159570 0.77 MAPT (0.32) CYP1A2
SCHEMBL8177031 0.76 ALDH1A1 (0.46) KDM4EKMT2A
SCHEMBL4611388 0.74 BRD4 (0.33) CYP1A2
SCHEMBL6543859 0.74 ALDH1A1 (0.49) KDM4E
SCHEMBL4612243 0.74 CA2 (0.44) CYP1A2CA2CHKAKMT2A
SCHEMBL1127702 0.74 ALDH1A1 (0.49) KDM4E
SCHEMBL7994140 0.74 CA2 (0.39) CYP1A2CA2CHKAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979319-A1 NOVEL DUAL NK2/NK3-ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND PROCESSES FOR THEIR PREPARATIONS Solvay Pharmaceuticals GmbH (DE) 2008-10-15 EP disclosed
WO-2007088181-A1 NOVEL DUAL NK2/NK3-ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND PROCESSES FOR THEIR PREPARATIONS SOLVAY PHARMACEUTICALS GMBH (DE) 2007-08-09 WO disclosed
WO-2005047253-A1 MELANOCORTIN RECEPTOR AGONISTS LG LIFE SCIENCES LTD. (KR) 2005-05-26 WO disclosed