SCHEMBL4611897

SCHEMBL4611897

OC(CN1CCN(CCc2ccccc2)CC1)c1ccncc1.c1ccc(CCN2CCN(CCCc3cccnc3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 1/20 0.51
ALOX15 P16050 1/20 0.51
SIGMAR1 Q99720 3/20 0.50
GAA P10253 1/20 0.45
PTAFR P25105 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4611120 0.89 KDM4E (0.49) KDM4EGAA
SCHEMBL4164330 0.89 KDM4E (0.58) KDM4EGAA
SCHEMBL4164304 0.85 KDM4E (0.55) KDM4EGAA
SCHEMBL4169559 0.85 SIGMAR1 (0.67) KDM4EALDH1A1ALOX15SIGMAR1
Bromide SCHEMBL4173363 0.84 KDM4E (0.53) KDM4EGAA
Bromide SCHEMBL4174825 0.83 SIGMAR1 (0.65) KDM4EALDH1A1ALOX15SIGMAR1
SCHEMBL4168265 0.79 SLC6A3 (0.59) SIGMAR1
Bromide SCHEMBL4171916 0.78 SLC6A3 (0.58) SIGMAR1
SCHEMBL4474652 0.78 KDM4E (0.74) KDM4EALDH1A1GAA
SCHEMBL11721357 0.74 GAA (0.56) KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981849-A1 HETEROCYCLIC COMPOUNDS LEK Pharmaceuticals D.D. (SI) 2008-10-22 EP claimed
WO-2007073935-A1 HETEROCYCLIC COMPOUNDS LEK PHARMACEUTICALS D.D. (SI) 2007-07-05 WO claimed