SCHEMBL4613355

SCHEMBL4613355

Nc1ncc(-c2ccccc2F)c(N)n1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.51
ADORA1 P30542 1/20 0.45
ALOX5AP P20292 2/20 0.44
FEN1 P39748 2/20 0.44
ADORA2A P29274 1/20 0.44
BCL6 P41182 1/20 0.44
NPC1 O15118 1/20 0.43
MPL P40238 1/20 0.43
USP7 Q93009 1/20 0.43
AURKA O14965 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12813395 0.82 CHRM5 (0.46) ADORA2ANPC1MPLUSP7
SCHEMBL27613072 0.78 DHFR (0.59) DHFRADORA1ADORA2A
SCHEMBL4464780 0.78 FGFR1 (0.55) DHFRADORA1ADORA2A
SCHEMBL28201122 0.78 DHFR (0.51) DHFR
SCHEMBL4186547 0.78 DHFR (0.56) DHFRADORA1ADORA2ABCL6
SCHEMBL15648676 0.78 ADORA2A (0.56) ADORA1ALOX5APFEN1ADORA2ABCL6
SCHEMBL29114862 0.77 DHFR (0.47) DHFRADORA1ALOX5APFEN1ADORA2A
SCHEMBL3959532 0.76 DHFR (0.54) DHFR
SCHEMBL27612436 0.76 DHFR (0.45) DHFRADORA1ALOX5APFEN1BCL6
SCHEMBL1612797 0.76 DHFR (0.45) DHFRADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981856-A2 PYRIMIDINE DERIVATIVES AstraZeneca AB (SE) 2008-10-22 EP disclosed
WO-2007085833-A2 PYRIMIDINE DERIVATIVES ASTRAZENECA AB (SE) 2007-08-02 WO disclosed